Elagolix sodiumCS-01Y78396_上海莼试生物技术有限公司

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一、概述：

化学性质：

规格	5mg 10mg 50mg 100mg
CAS	832720-36-2
别名	N/A
化学名	N/A
分子式	C32H29F5N3NaO5
分子量	653.57
溶解度	DMSO : 50 mg/mL (76.50 mM);H2O : ≥ 50 mg/mL (76.50 mM)
储存条件	Store at -20°C
General tips	For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition	Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request

产品描述：

Elagolix sodium is a human GnRH receptor (GnRHR) antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.

Elagolix sodium is a human GnRH receptor (GnRHR) antagonist with an IC50 of 0.25 nM in Kinase assay. Elagolix sodium has advanced to phase 3 trials for the treatment of endometriosis and uterine fibroids. Elagolix sodium also shows NFAT inhibition with an IC50 of 5.4 nM and effectively blocks Ca2+ flux with an IC50 of 0.86 nM[1]. Kinase assay also demonstrates that Elagolix sodium is a human GnRH receptor (GnRHR) antagonist with a Ki value of 3.7 nM[2].

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标签：Elagolix sodium

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