Sigma-1 receptor antagonist 3CS-01Y75346_上海莼试生物技术有限公司

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一、概述：

化学性质：

规格	1mg 5mg 10mg 50mg 100mg
CAS	1639220-17-9
别名	N/A
化学名	N/A
分子式	C19H23ClFN3O
分子量	363.86
溶解度	DMSO: 12.5 mg/mL (34.35 mM)
储存条件	Store at -20°C
General tips	For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition	Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request

产品描述：

Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 μM. Sigma-1 receptor antagonist 3 is for treating neuropathic pain[1].

[1]. Lan Y, et al. Synthesis and biological evaluation of novel sigma-1 receptor antagonists based on pyrimidine scaffold as agents for treating neuropathic pain. J Med Chem. 2014 Dec 26;57(24):10404-23.

特别提醒：

1. 本产品仅供科研使用。请勿用于医药、临床诊断或治疗，食品及化妆品等用途。请勿存放于普通住宅区。

2. 为了您的安全和健康，请穿好实验服并佩戴一次性手套和口罩操作。

标签：Sigma-1 receptor antagonist 3

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抑制剂 > 膜转运蛋白/离子通道 > Sigma-1 receptor antagonist 3

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